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dBET57

Glpbio
Catalog No:GC35815-10mM (in 1mL DMSO) CAS No.:1883863-52-2 MDLNo: Brand:Glpbio purity: 特性: Purpose:dBET57 是一种有效选择性的 BRD4BD1 降解剂,基于 PROTAC 技术。dBET57 介导了 E3 泛素连接酶 CRL4CRBN 的招募,对 BRD4BD1 作用的 DC50/5h 值为 500 nM,对 BRD4BD2 不起作用。DMSO: 250 mg/mL (357.56 mM)
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